{"id":21786,"date":"2020-04-23T00:00:45","date_gmt":"2020-04-22T16:00:45","guid":{"rendered":"https:\/newsletter.sinica.edu.tw\/?p=21786"},"modified":"2021-09-30T11:52:58","modified_gmt":"2021-09-30T03:52:58","slug":"%e3%80%90%e4%b8%ad%e7%a0%94%e6%8a%97%e7%96%ab2%e3%80%91%e5%b0%8f%e5%88%86%e5%ad%90%e8%97%a5%e7%89%a9%e7%a0%94%e7%99%bc%e7%ad%96%e7%95%a5%ef%bc%9a%e5%84%aa%e5%85%88%e8%80%83%e6%85%ae%e5%ad%b8%e5%90%8d","status":"publish","type":"post","link":"https:\/newsletter.sinica.edu.tw\/21786\/","title":{"rendered":"\u3010\u4e2d\u7814\u6297\u75ab2\u3011\u5c0f\u5206\u5b50\u85e5\u7269\u7814\u767c\u7b56\u7565\uff1a\u512a\u5148\u8003\u616e\u5b78\u540d\u85e5\uff0c\u76fc\u53ca\u6642\u627e\u5230\u6551\u547d\u89e3\u65b9"},"content":{"rendered":"

\u4e2d\u7814\u9662\u65b0\u51a0\u80ba\u708e\u5c0f\u5206\u5b50\u85e5\u7269\u7814\u767c<\/strong><\/h1>\n

\u4e16\u754c\u885b\u751f\u7d44\u7e54\uff08WHO\uff09\u79d8\u66f8\u9577\u8b5a\u5fb7\u585e\u5df2\u5728 3 \u6708 11 \u865f\uff0c\u5ba3\u5e03\u65b0\u578b\u51a0\u72c0\u75c5\u6bd2\u75ab\u60c5\u9032\u5165\u300c\u5168\u7403\u5927\u6d41\u884c\uff08pandemic\uff09\u300d\uff0c\u5404\u79d1\u6280\u5927\u570b\u6b63\u5982\u706b\u5982\u837c\u5730\u7814\u767c\u7279\u6548\u85e5\u7269\u3002\u4e2d\u7814\u9662\u751f\u91ab\u8f49\u8b6f\u7814\u7a76\u4e2d\u5fc3\u526f\u4e3b\u4efb\u8b1d\u8208\u90a6\u6307\u51fa\uff0c\u9662\u5167\u5df2\u6210\u7acb\u6297\u75c5\u6bd2\u5c0f\u5206\u5b50\u85e5\u7269\u7814\u7a76\u5c0f\u7d44\uff0c\u8207\u570b\u5167\u5404\u7814\u7a76\u55ae\u4f4d\u5171\u5275\u85e5\u7269\u8cc7\u6e90\u5171\u4eab\u5e73\u53f0\uff0c\u63a1\u53d6\u300c\u8001\u85e5\u65b0\u7528\u300d\u7b56\u7565\uff0c\u5f9e\u5065\u4fdd\u5b78\u540d\u85e5\u4e0b\u624b\uff0c\u4ee5\u671f\u76e1\u901f\u627e\u5230\u6709\u6548\u85e5\u7269\u3002<\/strong><\/p>\n

<\/p>\n

\u4eca\u5e74 (2020\u5e74) 2 \u6708\uff0c\u4e2d\u7814\u9662\u5316\u5b78\u6240\u9673\u69ae\u5091\u526f\u7814\u7a76\u54e1\u5718\u968a\uff0c\u6210\u529f\u5408\u6210\u300c\u767e\u6beb\u514b\u7d1a\u300d\u3001\u7d14\u5ea6\u9054\u767e\u5206\u4e4b 97 \u7684\u745e\u5fb7\u897f\u97cb\uff0c\u4e14\u5df2\u7cbe\u9032\u5230\u300c\u516c\u514b\u7d1a\u300d\u3001\u7d14\u5ea6 99%\u3002\u6d88\u606f\u4e00\u51fa\uff0c\u5f15\u7206\u5168\u81fa\u71b1\u8b70\uff0c\u56e0\u70ba\u745e\u5fb7\u897f\u97cb (Remdesivir) \u70ba\u7576\u524d\u6700\u6709\u5e0c\u671b\u5c0d\u6297\u65b0\u51a0\u80ba\u708e\u7684\u5019\u9078\u85e5\u7269\u3002<\/p>\n

\u6839\u64da 4 \u6708 11 \u65e5\u300c\u65b0\u82f1\u683c\u862d\u91ab\u5b78\u671f\u520a\u300d(New England Journal of Medicine) \u7684\u6700\u65b0\u7814\u7a76\uff0c\u4f86\u81ea\u7f8e\u570b\u548c\u5168\u7403\u7684 53 \u540d\u75c5\u60a3\u900f\u904e\u6069\u6148\u7642\u6cd5\uff0c\u63a5\u53d7\u745e\u5fb7\u897f\u97cb\u6cbb\u7642\u5f8c\uff0c\u4e09\u5206\u4e4b\u4e8c\u60a3\u8005\u7684\u75c5\u60c5\u7372\u5f97\u7de9\u89e3\uff0c\u70ba\u5168\u7403\u885b\u751f\u7576\u5c40\u5e36\u4f86\u6b63\u9762\u6d88\u606f\uff0c\u4f46\u4ecd\u9700\u8981\u7b49\u5f85\u63a7\u5236\u5b89\u6170\u5291\u7684\u96d9\u76f2\u8a66\u9a57\u7d50\u679c\uff0c\u624d\u80fd\u78ba\u8a8d\u745e\u5fb7\u897f\u97cb\u7684\u7642\u6548\u3002\u6545\u6b64\uff0c\u5168\u7403\u79d1\u7814\u55ae\u4f4d\u7686\u540c\u6b65\u5c0b\u627e\u66f4\u591a\u53ef\u80fd\u5099\u9078\u85e5\u7269\uff0c\u81fa\u7063\u81ea\u4e0d\u4f8b\u5916\u3002<\/p>\n

\u53ea\u662f\u5f9e\u96f6\u7814\u767c\u65b0\u85e5\u7de9\u4e0d\u6fdf\u6025\uff0c\u4e2d\u7814\u9662\u65b0\u51a0\u80ba\u708e\u6297\u75c5\u6bd2\u5c0f\u5206\u5b50\u85e5\u7269\u5c0f\u7d44\u53ec\u96c6\u4eba\u2014\u2014\u8b1d\u8208\u90a6\u7814\u7a76\u54e1\u517c\u526f\u4e3b\u4efb\uff0c\u64ec\u5b9a\u300c\u8001\u85e5\u65b0\u7528\u300d\u3001\u958b\u767c\u5065\u4fdd\u5b78\u540d\u85e5\u7b49\u7b56\u7565\uff0c\u671f\u5f85\u5f9e\u904e\u53bb\u85e5\u7269\u53ca\u6642\u627e\u5230\u6709\u6548\u89e3\u65b9\u3002\u4eca\u5e74 (2020 \u5e74) 4 \u6708 10 \u65e5\u50b3\u51fa\u521d\u6b65\u6377\u5831 \uff0c\u751f\u7269\u5316\u5b78\u7814\u7a76\u6240\u6881\u535a\u714c\u7814\u7a76\u54e1\u5f9e\u4e0a\u767e\u7a2e\u5316\u5408\u7269\u4e2d\u7be9\u9078\u51fa\u65b0\u51a0\u75c5\u6bd2\u985e\u86cb\u767d\u9176\u6291\u5236\u5291\uff0c\u5df2\u8b49\u5be6\u53ef\u5728\u9ad4\u5916\u6291\u5236\u65b0\u51a0\u75c5\u6bd2\u8907\u88fd\u3002<\/p>\n

\"\u4e2d\u7814\u9662\u751f\u91ab\u8f49\u8b6f\u7814\u7a76\u4e2d\u5fc3\u8b1d\u8208\u90a6\u526f\u4e3b\u4efb\uff0c\u65bc\u672c\u6b21\u4e2d\u7814\u9662\u65b0\u51a0\u80ba\u708e\u6297\u75c5\u6bd2\u5c0f\u5206\u5b50\u85e5\u7269\u5c0f\u7d44\u64d4\u4efb\u53ec\u96c6\u4eba\uff0c\u64ec\u5b9a\u8001\u85e5\u65b0\u7528\u3001\u5065\u4fdd\u5b78\u540d\u85e5\u512a\u5148\u7b49\u91cd\u8981\u7b56\u7565\u3002\u651d\u5f71\u2502\u6797\u6d35\u5b89\"

\u4e2d\u7814\u9662\u751f\u91ab\u8f49\u8b6f\u7814\u7a76\u4e2d\u5fc3\u8b1d\u8208\u90a6\u526f\u4e3b\u4efb\uff0c\u65bc\u672c\u6b21\u4e2d\u7814\u9662\u65b0\u51a0\u80ba\u708e\u6297\u75c5\u6bd2\u5c0f\u5206\u5b50\u85e5\u7269\u5c0f\u7d44\u64d4\u4efb\u53ec\u96c6\u4eba\uff0c\u64ec\u5b9a\u8001\u85e5\u65b0\u7528\u3001\u5065\u4fdd\u5b78\u540d\u85e5\u512a\u5148\u7b49\u91cd\u8981\u7b56\u7565\u3002 \u651d\u5f71\u2502\u6797\u6d35\u5b89<\/p><\/div>\n

 <\/p>\n

\u7814\u767c\u85e5\u7269\uff0c\u5f9e\u9776\u9ede\u958b\u59cb<\/b><\/strong><\/h2>\n

\u4e0d\u8ad6\u5f9e\u96f6\u958b\u59cb\u6216\u8001\u85e5\u65b0\u7528\uff0c\u7814\u767c\u6297\u75c5\u6bd2\u85e5\u7269\u7684\u95dc\u9375\u70ba\uff1a\u627e\u5230\u6291\u5236\u75c5\u6bd2\u8907\u88fd\u7684\u5206\u5b50\u6216\u5316\u5408\u7269\uff0c\u4f5c\u70ba\u85e5\u7269\u7684\u539f\u6599\u2014-\u5148\u5c0e\u85e5\u7269<\/a>\uff08lead compound\uff09\u3002\u4f46\u5c0b\u627e\u5148\u5c0e\u85e5\u7269\u4e26\u975e\u4e82\u69cd\u6253\u9ce5\uff0c\u4e00\u958b\u59cb\u5fc5\u9808\u5148\u9078\u64c7\u7279\u5b9a\u7684\u300c\u9776\u9ede<\/a>\u300d\u3002<\/p>\n

\u300c\u9776\u9ede\u300d\uff0c\u5373\u662f\u85e5\u7269\u5206\u5b50\u4f5c\u7528\u7684\u76ee\u6a19\uff0c\u901a\u5e38\u662f\u6307\u4ee5\u85e5\u7269\u5e72\u64fe\u300c\u75c5\u6bd2\u8907\u88fd\u904e\u7a0b\u7684\u67d0\u500b\u968e\u6bb5\u300d\uff0c\u76ee\u7684\u662f\u7a69\u5b9a\u3001\u6709\u6548\u5730\u58d3\u5236\u75c5\u6bd2\u3002\u8b1d\u8208\u90a6\u6bd4\u55bb\uff0c\u75c5\u6bd2\u5165\u4fb5\u7d30\u80de\u5c31\u50cf\u5c0f\u7de8\u8d70\u9032\u4e2d\u7814\u9662\u751f\u91ab\u8f49\u8b6f\u4e2d\u5fc3\uff0c\u5fc5\u9808\u901a\u904e\u5c64\u5c64\u95dc\u5361\u6aa2\u67e5\u3002\u53ea\u8981\u5176\u4e2d\u4e00\u9053\u95dc\u5361\u64cb\u4f4f\u4e86\uff0c\u5c0f\u7de8 (\u75c5\u6bd2) \u5c31\u7121\u6cd5\u5b8c\u6210\u4efb\u52d9\u4e86\u3002<\/p>\n

\n

\u5f9e\u75c5\u6bd2\u8907\u88fd\u904e\u7a0b\uff0c\u627e\u51fa\u5b83\u7684\u963f\u57fa\u91cc\u65af\u8171\u3002<\/strong><\/h4>\n<\/blockquote>\n

\u4ee5\u65b0\u578b\u51a0\u72c0\u75c5\u6bd2\u6240\u5c6c\u7684\u6838\u7cd6\u6838\u9178\uff08ribonucleic acid, RNA\uff09\u75c5\u6bd2\u4f86\u8aaa\uff0c\u75c5\u6bd2\u85c9\u7531\u80de\u541e\u4f5c\u7528\uff08endocytosis\uff09\u9032\u5165\u7d30\u80de\u5f8c\uff0c\u6703\u5148\u5c07\u81ea\u5df1\u5206\u89e3\u3001\u628a\u907a\u50b3\u7269\u8cea\uff08RNA\uff09\u91cb\u653e\u51fa\u4f86\uff0c\u4ee5\u5229\u8907\u88fd\u3002\u63a5\u8457\uff0c\u75c5\u6bd2\u6703\u5f37\u8feb\u5bbf\u4e3b\u7d30\u80de\u7684\u86cb\u767d\u8cea\u5408\u6210\u7cfb\u7d71\uff0c\u6309\u7167\u75c5\u6bd2\u4fe1\u4f7f RNA\uff08messenger RNA, mRNA\uff09\uff0c\u5408\u6210\u75c5\u6bd2\u8907\u88fd\u6240\u9700\u7684\u86cb\u767d\u8cea\u300c\u96f6\u4ef6\u300d\u8207 RNA\u3002\u9019\u4e9b\u86cb\u767d\u8cea\u300c\u96f6\u4ef6\u300d\u548c RNA \u6703\u91cd\u65b0\u7d44\u88dd\u6210\u6578\u767e\u500b\u5b8c\u6574\u65b0\u75c5\u6bd2\uff0c\u6700\u5f8c\u96e2\u958b\u5bbf\u4e3b\u7d30\u80de\u3002<\/p>\n

\u9776\u9ede\u5728\u54ea\uff1f\u6bd4\u65b9\u8aaa\uff1a\u5728\u75c5\u6bd2\u8907\u88fd\u904e\u7a0b\u4e2d\uff0c\u662f\u7531\u8a31\u591a\u86cb\u767d\u9176<\/a>\uff08enzyme\uff09\u8ca0\u8cac\u75c5\u6bd2\u86cb\u767d\u8cea\u548c RNA \u7684\u5408\u6210\u3001\u5207\u5272\u3001\u91cd\u7d44\u7b49\u7b49\u5de5\u4f5c\u3002\u53ea\u8981\u60f3\u8fa6\u6cd5\u6291\u5236\u9019\u4e9b\u86cb\u767d\u9176\u7684\u6d3b\u6027\uff0c\u5c31\u53ef\u4ee5\u9054\u5230\u300c\u5361\u95dc\u300d\u7684\u76ee\u7684\u3002\u4e00\u822c\u4f86\u8aaa\uff0c\u4ee5\u6b3a\u6575\u6230\u7565\u5c45\u591a\uff0c\u4e5f\u5c31\u662f\u4f7f\u7528\u5316\u5b78\u7d50\u69cb\u76f8\u4f3c\u7684\u5206\u5b50\u4f86\u4ee3\u66ff\u5408\u6210\u6642\u6240\u9700\u8981\u7684\u300c\u96f6\u4ef6\u300d\uff0c\u5373\u6709\u6a5f\u6703\u963b\u65b7\u8907\u88fd\u6d41\u7a0b\uff0c\u800c\u9019\u4e9b\u53ef\u88ab\u77c7\u9a19\u7684\u86cb\u767d\u9176\u5c31\u6210\u70ba\u5f88\u597d\u7684\u9776\u9ede\u3002<\/p>\n

\u62ff\u8457\u540d\u7684\u5019\u9078\u85e5\u7269\u745e\u5fb7\u897f\u97cb\u800c\u8a00\uff0c\u5373\u4ee5\u75c5\u6bd2 RNA \u8907\u88fd\u6240\u9700\u00a0RdRp \u805a\u5408\u9176<\/a>\uff08RNA-dependent RNA polymerase, RdRp\uff09\u70ba\u9776\u9ede\uff0c\u7528\u745e\u5fb7\u897f\u97cb\u7684\u5206\u5b50\u5192\u5145\u75c5\u6bd2 RNA \u7684\u96f6\u4ef6\uff0c\u6b3a\u9a19 RdRp \u805a\u5408\u9176\u62ff\u5b83\u53bb\u7d44\u88dd\u65b0\u7684 RNA\uff0c\u4f7f\u7d44\u88dd\u5b8c\u6210\u7684 RNA \u5b9b\u5982\u88ab\u585e\u5165\u7570\u7269\u7684\u6a5f\u5668\uff0c\u7121\u6cd5\u767c\u63ee\u6b63\u5e38\u529f\u80fd\u3002<\/p>\n

 <\/p>\n

\"(1a)\u75c5\u6bd2\u68d8\u86cb\u767d\u8207\u7d30\u80de\u8868\u9762\u53d7\u9ad4

(1a)\u75c5\u6bd2\u68d8\u86cb\u767d\u8207\u7d30\u80de\u8868\u9762\u53d7\u9ad4 ACE2 \u7d50\u5408\uff0c\u5c31\u50cf\u7528\u9396\u63d2\u5165\u9470\u5319\u958b\u9580\uff0cTMPRSS2 \u5247\u6703\u5e6b\u52a9\u75c5\u6bd2\u9032\u5165\u7d30\u80de\u3002 (1b)\u7d30\u80de\u819c\u51f9\u9677\u5f62\u6210\u56ca\u6ce1\uff0c\u628a\u75c5\u6bd2\u5305\u88f9\u8d77\u4f86\uff0c\u9032\u5165\u7d30\u80de\u3002 (2) \u75c5\u6bd2\u9032\u5165\u7d30\u80de\u5f8c\u6703\u91cb\u653e\u907a\u50b3\u7269\u8cea RNA \uff0c\u4e26\u5207\u65b7 RNA \u4ee5\u5229\u8907\u88fd\u3002 (3) \u75c5\u6bd2\u7d81\u67b6\u7d30\u80de\u7684\u86cb\u767d\u8cea\u5408\u6210\u7cfb\u7d71\uff0c\u88fd\u9020\u75c5\u6bd2\u8907\u88fd\u6240\u9700\u5404\u7a2e\u591a\u80dc\u80bd\u3002 (4) \u6709\u4e9b\u591a\u80dc\u80bd\u8ca0\u8cac\u8907\u88fd\u75c5\u6bd2 RNA\uff0c\u6709\u4e9b\u8907\u88fd\u75c5\u6bd2\u7d50\u69cb\u7684\u300c\u5143\u4ef6\u300d\u3002 (5) \u5c07\u8907\u88fd\u5b8c\u6210\u7684 RNA \u8207\u7d50\u69cb\u5143\u4ef6\uff0c\u7d44\u5408\u6210\u4e00\u500b\u500b\u65b0\u75c5\u6bd2 \u3002 (6) \u65b0\u75c5\u6bd2\u96e2\u958b\u5bbf\u4e3b\u7d30\u80de\u3002 \u8cc7\u6599\u4f86\u6e90\u2502\u8b1d\u8208\u90a6 \u5716\u8aaa\u91cd\u88fd\u2502\u9ec3\u66c9\u541b\u3001\u6797\u6d35\u5b89<\/p><\/div>\n

 <\/p>\n

 <\/p>\n

\u65b0\u85e5\u7814\u767c\uff1a\u5341\u5e74\u78e8\u4e00\u528d\u7684\u9ad8\u98a8\u96aa\u8ced\u6ce8<\/b><\/strong><\/h2>\n

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 <\/p>\n

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https:\/research.sinica.edu.tw\/covid-19-drug-academia-sinica\/<\/em><\/a><\/h2>\n

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